Found 8 of kd for NOCICEPTIN RECEPTORhaving polymerids = 2210,49000818,49000820,49000821,49000886,50003607 and
complexids = 50002056
Affinity DataKd: 1.95nMAssay Description:Antagonist activity at NOR in mouse Neuro-2a cells assessed as inhibition of nociceptin-induced ERK phopshorylation administered for 15 mins before n...More data for this Ligand-Target Pair
Affinity DataKd: 0.100nMAssay Description:Compound was tested for inhibition against binding of radioligand [leucyl-3H]-OFQ to membrane of human embryonic kidney 293 cells overexpressing rat ...More data for this Ligand-Target Pair
Affinity DataKd: 0.190nMAssay Description:Binding affinity to human ORL1 receptor expressed in African green monkey COS7 cells assessed per mg protein after 90 mins by Scatchard plot analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0.794nMAssay Description:Antagonist activity at NOP receptor in Swiss mouse vas deferens by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.0920nMAssay Description:Binding affinity to recombinant ORL1 receptor expressed in COS7 cells by saturation binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.316nMAssay Description:Antagonist activity at NOP receptor in Albino guinea pig ileum assessed as effect on electrically stimulated contractionsMore data for this Ligand-Target Pair
Affinity DataKd: 0.603nMAssay Description:Antagonist activity at NOP receptor in Sprague-Dawley rat vas deferens assessed as effect on electrically stimulated contractionsMore data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Binding affinity to human ORL1 receptor expressed in African green monkey COS7 cells assessed per mg protein after 90 mins by Scatchard plot analysisMore data for this Ligand-Target Pair
